Oshitari Tetsuta

Researcher Information

Affiliation

Faculty of Pharmaceutical Sciences Professor

Degree

• Ph. D.（1995/03 The University of Tokyo）

URL

https://jglobal.jst.go.jp/detail?JGLOBAL_ID=200901081634526372

J-Global ID

• 200901081634526372

Research Interests

• 医薬品化学   有機合成化学   有機化学   Pharmaceutical Synthetic Chemistry   Synthetic Chemistry   Organic Chemistry   

Research Areas

• Life sciences / Pharmaceuticals - chemistry and drug development

Academic & Professional Experience

• 2015/04 - Today  Teikyo University
• 2008/04 - 2015/03  Teikyo UniversityFaculty of Pharma-Science
• 2004/04 - 2008/03  Kurashiki University of Science and the ArtsCollege of Life Science
• 1999/04 - 2004/03  Kurashiki University of Science and the ArtsCollege of Science and Industrial Technology
• 1995/04 - 1999/03  Kurashiki University of Science and the ArtsCollege of Science and Industrial Technology

Education

•        - 1990/03  The University of Tokyo  Faculty of Pharmaceutical Sciences  Department of Pharmacy

Association Memberships

• アメリカ化学会   有機合成化学協会   日本化学会   日本薬学会   

Research Activity Information

Published Papers

• Stereochemistry of N-Acyl-5H-dibenzo[b,d]azepin-7(6H)-ones

  Arisa Chiba; Ryoko Tanaka; Mayuno Hotta; Kayo Nakamura; Kosho Makino; Hidetsugu Tabata; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  Molecules MDPI AG 28 (12) 4734 - 4734 2023/06
• Stereochemical Analysis of Trifluoroacetamide Derivatives Based on Through-Space ¹H–¹⁹F Spin–Spin Couplings

  Yan Li; Chinatsu Ohtake; Mayuno Hotta; Hidetsugu Tabata; Kiriko Hirano; Motoo Iida; Kayo Nakamura; Kosho Makino; Tetsuta Oshitari; Hideaki Natsugari; Takenori Kusumi; Hideyo Takahashi

  The Journal of Organic Chemistry American Chemical Society (ACS) 88 (11) 7026 - 7037 0022-3263 2023/05
• Conversion of Racemic Alkyl Aryl Sulfoxides into Pure Enantiomers Using a Recycle Photoreactor: Tandem Use of Chromatography on Chiral Support and Photoracemization on Solid Support

  Kumi Tozawa; Kosho Makino; Yuki Tanaka; Kayo Nakamura; Akiko Inagaki; Hidetsugu Tabata; Tetsuta Oshitari; Hideaki Natsugari; Noritaka Kuroda; Kunio Kanemaru; Yuji Oda; Hideyo Takahashi

  The Journal of Organic Chemistry American Chemical Society (ACS) 0022-3263 2023/05
• Atropodiastereoselective 5N-Acylation of 1,5-Benzodiazepin-2-ones with (S)-2-Phenylpropanoyl and (S)-2-Phenylbutanoyl Chlorides

  Kaoru Funaki; Hidetsugu Tabata; Yusuke Nakazato; Yuka Takahashi; Tomohiko Tasaka; Hideyo Takahashi; Hideaki Natsugari; Tetsuta Oshitari

  The Journal of Organic Chemistry 87 (22) 15289 - 15300 2022/11 [Refereed]
  
• ノビレチンによるマウス褐色脂肪細胞の熱産生およびブラウンアディポカイン分泌促進の機構解析

  根岸 文子; 大藏 直樹; 高橋 由佳; 中村 康宏; 丸山 桂司; 忍足 鉄太

  日本生化学会大会プログラム・講演要旨集 (公社)日本生化学会 95回 1P - 277 2022/11
• Atropisomeric Properties of N-Alkyl/Aryl 5H-Dibenz[b,f]azepines

  Ryoko Tanaka; Ayana Nabae; Koki Yamane; Kosho Makino; Hidetsugu Tabata; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  Chemical and Pharmaceutical Bulletin Pharmaceutical Society of Japan 70 (8) 573 - 579 0009-2363 2022/08 [Refereed]
  
• Axial chirality and affinity at the GABAA receptor of triazolobenzodiazepines

  Ryoko Tanaka; Kosho Makino; Hidetsugu Tabata; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  Bioorganic & Medicinal Chemistry Elsevier BV 64 116758 - 116758 0968-0896 2022/06 [Refereed]
  
• Nobiletin and 3′-Demethyl Nobiletin Activate Brown Adipocytes upon β-Adrenergic Stimulation

  Fumiko Kihara-Negishi; Naoki Ohkura; Yuka Takahashi; Toshiyuki Fujita; Yasuhiro Nakamura; Keiji Maruyama; Tetsuta Oshitari; Shinji Yamaguchi

  Biological and Pharmaceutical Bulletin Pharmaceutical Society of Japan 45 (4) 528 - 533 0918-6158 2022/04 [Refereed]
  
• Photoisomerization of Sulindac and Ozagrel Hydrochloride by Vitamin B2 Catalyst Under Visible Light Irradiation

  Mayuko Suga; Kosho Makino; Hidetsugu Tabata; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  Pharmaceutical Research Springer Science and Business Media LLC 39 (3) 577 - 586 0724-8741 2022/03 [Refereed]
  
• Rapid Photoracemization of Chiral Alkyl Aryl Sulfoxides

  Kosho Makino; Kumi Tozawa; Yuki Tanaka; Akiko Inagaki; Hidetsugu Tabata; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  The Journal of Organic Chemistry American Chemical Society (ACS) 86 (23) 17249 - 17256 0022-3263 2021/12 [Refereed]
  
• Atropisomeric Properties of 9-Methyl-1,4-benzodiazepin-2-ones

  Hideyo Takahashi; Ryoko Tanaka; Kosho Makino; Hidetsugu Tabata; Tetsuta Oshitari; Hideaki Natsugari

  Synthesis Georg Thieme Verlag KG 53 (24) 4682 - 4688 0039-7881 2021/12 [Refereed]
  
• Atropisomeric Properties of N-Acyl/N-Sulfonyl 5H-Dibenzo[b,d]azepin-7(6H)-ones

  Takuya Namba; Mayuno Hotta; Hidetsugu Tabata; Kosho Makino; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  The Journal of Organic Chemistry American Chemical Society (ACS) 86 (11) 7563 - 7578 0022-3263 2021/06 [Refereed]
  
• Conformational Preference of 2′-Fluoro-Substituted Acetophenone Derivatives Revealed by Through-Space 1H–19F and 13C–19F Spin–Spin Couplings

  Chinatsu Otake; Takuya Namba; Hidetsugu Tabata; Kosho Makino; Kiriko Hirano; Tetsuta Oshitari; Hideaki Natsugari; Takenori Kusumi; Hideyo Takahashi

  The Journal of Organic Chemistry American Chemical Society (ACS) 86 (6) 4638 - 4645 0022-3263 2021/03 [Refereed]
  
• Structural Requirements for Uptake of Diphenhydramine Analogs into hCMEC/D3 Cells Via the Proton-Coupled Organic Cation Antiporter

  Yuma Tega; Hidetsugu Tabata; Toshiki Kurosawa; Atsushi Kitamura; Fumio Itagaki; Tetsuta Oshitari; Yoshiharu Deguchi

  Journal of Pharmaceutical Sciences Elsevier BV 110 (1) 397 - 403 0022-3549 2021/01 [Refereed]
  
• Conformational properties and M1 antimuscarinic activity of 4-substituted pirenzepine/telenzepine analogues

  Kanase, Yuki; Makino, Kosho; Yoshinaga, Takashi; Tabata, Hidetsugu; Oshitari, Tetsuta; Natsugari, Hideaki; Takahashi, Hideyo

  Heterocycles 101 (1) 273 - 283 2019/08 [Refereed]
  
• Elucidation of the Active Conformation of Antiproliferative Sulfonamides, 5N‑Arylsulfonyl-1,5-benzodiazepin-2-ones

  Hidetsugu Tabata; Kaoru Funaki; Tomohiko Tasaka; Tetsuta Oshitari; Hideyo Takahashi; Hideaki Natsugari

  Journal of Organic Chemistry 84 16338 - 16345 2019 [Refereed]
  
• Atropisomeric and conformational properties of 6N-benzoyl- and 6N-p-tosyl-1,6-benzodiazocines: comparison with those of 1,5-benzodiazepines

  Hidetsugu Tabata; Kazuya Murai; Kaoru Funaki; Chihiro Takemae; Tomohiko Tasaka; Tetsuta Oshitari; Hideyo Takahashi; Hideaki Natsugari

  Heterocycles 99 (1) 566 - 581 2019/01 [Refereed]
  
• Chemoselective Demethylation of Methoxypyridine

  Makino, Kosho; Hasegawa, Yumi; Inoue, Takahide; Araki, Koji; Tabata, Hidetsugu; Oshitari, Tetsuta; Ito, Kiyomi; Natsugari, Hideaki; Takahashi, Hideyo

  Synlett Georg Thieme Verlag KG 30 (8) 951 - 954 0936-5214 2019 [Refereed]
  
• Atropisomerism in the 2,​3,​4,​5-​Tetrahydro-​1 H -​1,​5-​benzodiazepine Nucleus: Effects of Central Chirality at C3 on the N-​Mesylation Reaction

  Tabata, Hidetsugu; Tsuji, Yuka; Yoneda, Tetsuya; Tasaka, Tomohiko; Oshitari, Tetsuta; Takahashi, Hideyo; Natsugari, Hideaki

  SYNLETT 29 (16) 2141 - 2146 2018/08 [Refereed]
  
• 4-Substituted carbamazepine derivatives: Conformational analysis and sodium channel-blocking properties

  Yuki Kanase; Takafumi Kitada; Hidetsugu Tabata; Kosho Makino; Tetsuta Oshitari; Hiromi Ohashi; Takashi Yoshinaga; Hideaki Natsugari; Hideyo Takahashi

  Bioorganic and Medicinal Chemistry Elsevier Ltd 26 (9) 2508 - 2513 1464-3391 2018/05 [Refereed]
  
• SYNTHESIS OF 3-AROYLINDOLES AS INTERMEDIATES OF CANNABIMIMETICS AND ELUCIDATION OF THEIR PHYSICOCHEMICAL PROPERTIES

  Araki Koji; Makino Kosho; Tabata Hidetsugu; Nakayama Hiroshi; Zaitsu Kei; Oshitari Tetsuta; Natsugari Hideaki; Takahashi Hideyo

  HETEROCYCLES 96 (5) 914 - 924 0385-5414 2018/05 [Refereed]
  
• 4-Substituted carbamazepine derivatives: Conformational analysis and sodium channel-blocking properties

  Kanase Yuki; Kitada Takafumi; Tabata Hidetsugu; Makino Kosho; Oshitari Tetsuta; Natsugari Hideaki; Ohashi Hiromi; Yoshinaga Takashi; Takahashi Hideyo

  Bioorganic & medicinal chemistry 26 (9) 2508 - 2513 0936-5214 2018 [Refereed]
  
• Elucidation of the E-Amide Preference of N-Acyl Azoles

  Yuka Takahashi; Hirotaka Ikeda; Yuki Kanase; Kosho Makino; Hidetsugu Tabata; Tetsuta Oshitari; Satoshi Inagaki; Yuko Otani; Hideaki Natsugari; Hideyo Takahashi; Tomohiko Ohwada

  JOURNAL OF ORGANIC CHEMISTRY AMER CHEMICAL SOC 82 (21) 11370 - 11382 0022-3263 2017/11 [Refereed]
  
• In vitro studies on nobiletin isolated from citrus plants and the bioactive metabolites, inhibitory action against gelatinase enzymatic activity and the molecular mechanisms in human retinal Muller cell line

  Yoshiki Miyata; Terumasa Nagase; Yoshiya Katsura; Hideyo Takahashi; Hideaki Natsugari; Tetsuta Oshitari; Hiroshi Kosano

  BIOMEDICINE & PHARMACOTHERAPY ELSEVIER FRANCE-EDITIONS SCIENTIFIQUES MEDICALES ELSEVIER 93 70 - 80 0753-3322 2017/09 [Refereed]
  
• Catalytic asymmetric S-oxidation of N-benzoyl-1,5-benzothiazepines

  Kosho Makino; Tetsuya Yoneda; Risa Ogawa; Yuki Kanase; Hidetsugu Tabata; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  TETRAHEDRON LETTERS PERGAMON-ELSEVIER SCIENCE LTD 58 (30) 2885 - 2888 0040-4039 2017/07 [Refereed]
  
• Tolvaptan-Type Vasopressin Receptor Ligands: Important Role of Axial Chirality in the Active Form

  Hidetsugu Tabata; Tetsuya Yoneda; Tetsuta Oshitari; Hideyo Takahashi; Hideaki Natsugari

  JOURNAL OF MEDICINAL CHEMISTRY AMER CHEMICAL SOC 60 (10) 4503 - 4509 0022-2623 2017/05 [Refereed]
  
• Electronic effects on the amide E-/Z-preference of N-benzoyl-carbazole derivatives

  Susumu Kayama; Norihiko Tani; Hidetsugu Tabata; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  TETRAHEDRON LETTERS PERGAMON-ELSEVIER SCIENCE LTD 57 (22) 2395 - 2398 0040-4039 2016/06 [Refereed]
  
• Stereochemistry of N-Benzoyl-5-substituted-1-benzazepines Revisited: Synthesis of the Conformationally Biased Derivatives and Revision of the Reported Structure

  Hidetsugu Tabata; Tetsuya Yoneda; Tomohiko Tasaka; Shigekazu Ito; Tetsuta Oshitari; Hideyo Takahashi; Hideaki Natsugari

  JOURNAL OF ORGANIC CHEMISTRY AMER CHEMICAL SOC 81 (8) 3136 - 3148 0022-3263 2016/04 [Refereed]
  
• Freezing the Butterfly Motion of Carbamazepine Derivatives

  Yuki Kanase; Mai Kuniyoshi; Hidetsugu Tabata; Yuka Takahashi; Susumu Kayama; Shintaro Wakamatsu; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  Synthesis (Germany) Georg Thieme Verlag 47 (24) 3907 - 3913 1437-210X 2015/12 [Refereed]
  
• Freezing the Butterfly Motion of Carbamazepine Derivatives

  Yuki Kanase; Mai Kuniyoshi; Hidetsugu Tabata; Yuka Takahashi; Susumu Kayama; Shintaro Wakamatsu; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  SYNTHESIS-STUTTGART GEORG THIEME VERLAG KG 47 (24) 3907 - 3913 0039-7881 2015/12 [Refereed]
  
• Stereochemical properties of N-benzoylated carbazole derivatives

  Susumu Kayama; Hidetsugu Tabata; Yuka Takahashi; Norihiko Tani; Shintaro Wakamatsu; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  TETRAHEDRON PERGAMON-ELSEVIER SCIENCE LTD 71 (38) 7046 - 7053 0040-4020 2015/09 [Refereed]
  
• Isolation of Atropisomers of N-Benzoylated Pyrroles and Imidazoles

  Yuka Takahashi; Shintaro Wakamatsu; Hidetsugu Tabata; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  SYNTHESIS-STUTTGART GEORG THIEME VERLAG KG 47 (14) 2125 - 2128 0039-7881 2015/07 [Refereed]
  
• N-Benzoyl-1,5-benzothiazepine and Its S-Oxide as Vasopressin Receptor Ligands: Insight into the Active Stereochemistry around the Seven-Membered Ring

  Tetsuya Yoneda; Hidetsugu Tabata; Tomohiko Tasaka; Tetsuta Oshitari; Hideyo Takahashi; Hideaki Natsugari

  JOURNAL OF MEDICINAL CHEMISTRY AMER CHEMICAL SOC 58 (7) 3268 - 3273 0022-2623 2015/04 [Refereed]
  
• Development of a Therapeutic Agent for Menkes Disease: Solubilization of a Copper-Disulfiram Complex

  Yujiro Hoshi; Norihiko Tani; Hidetsugu Tabata; Shintaro Wakamatsu; Mitsutoshi Munakata; Kazuo Maruyama; Hiroko Kodama; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  YAKUGAKU ZASSHI-JOURNAL OF THE PHARMACEUTICAL SOCIETY OF JAPAN PHARMACEUTICAL SOC JAPAN 135 (3) 493 - 499 0031-6903 2015/03 [Refereed]
  
• Crystallization-Induced Diastereomeric Transformation of N-2'-t-Butyl-6'-iodobenzoyl-3-bromocarbazole

  Susumu Kayama; Norihiko Tani; Yuka Takahashi; Hidetsugu Tabata; Shintaro Wakamatsu; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  CHEMICAL & PHARMACEUTICAL BULLETIN PHARMACEUTICAL SOC JAPAN 62 (8) 836 - 838 0009-2363 2014/08 [Refereed]
  
• N-Benzoyl- and N-Sulfonyl-1,5-benzodiazepines: Comparison of Their Atropisomeric and Conformational Properties

  Tetsuya Yoneda; Hidetsugu Tabata; Jun Nakagomi; Tomohiko Tasaka; Tetsuta Oshitari; Hideyo Takahashi; Hideaki Natsugari

  JOURNAL OF ORGANIC CHEMISTRY AMER CHEMICAL SOC 79 (12) 5717 - 5727 0022-3263 2014/06 [Refereed]
  
• A Complete Gear System in N-Benzoyl-Carbazole Derivatives

  Hidetsugu Tabata; Susumu Kayama; Yuka Takahashi; Norihiko Tani; Shintaro Wakamatsu; Tomohiko Tasaka; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  ORGANIC LETTERS AMER CHEMICAL SOC 16 (5) 1514 - 1517 1523-7060 2014/03 [Refereed]
  
• Incompativility between Meropenem Injection and Amino Acid Infusions caused by L-Cysteine

  Itagaki F; KUdo, C; Katagiri S; Oshitari T; Takahashi H; Natsugari H; Watanabe M

  Japanese Journal of Pharmaceutical Health Care and Sciences Japanese Society of Pharmaceutical Health Care and Sciences 39 (9) 521 - 527 1346-342X 2013/09 [Refereed]
  
• Stereochemistry of 1,5-Benzothiazepin-4-one S-Oxide: Insight into the Stereogenic Elements at the Sulfur Atom and Axis

  Hidetsugu Tabata; Tetsuya Yoneda; Tetsuta Oshitari; Hideyo Takahashi; Hideaki Natsugari

  JOURNAL OF ORGANIC CHEMISTRY AMER CHEMICAL SOC 78 (12) 6264 - 6270 0022-3263 2013/06 [Refereed]
  
• Conformation and atropisomeric properties of indometacin derivatives

  Shintaro Wakamatsu; Yuka Takahashi; Hidetsugu Tabata; Tetsuta Oshitari; Norihiko Tani; Isao Azumaya; Yukiteru Katsumoto; Takeyuki Tanaka; Shinzo Hosoi; Hideaki Natsugari; Hideyo Takahashi

  Chemistry - A European Journal 22 19 (22) 7056 - 7063 0947-6539 2013/05 [Refereed]
  
• Polymethoxyflavones as agents that prevent formation of cataract: Nobiletin congeners show potent growth inhibitory effects in human lens epithelial cells

  Yoshiki Miyata; Tetsuta Oshitari; Yuji Okuyama; Arata Shimada; Hideyo Takahashi; Hideaki Natsugari; Hiroshi Kosano

  BIOORGANIC & MEDICINAL CHEMISTRY LETTERS PERGAMON-ELSEVIER SCIENCE LTD 23 (1) 183 - 187 0960-894X 2013/01 [Refereed]
  
• Active Conformation of Seven-Membered-Ring Benzolactams as New ACAT Inhibitors: Latent Chirality at N5 in the 1,5-Benzodiazepin-2-one Nucleus

  Hidetsugu Tabata; Naoya Wada; Yuko Takada; Jun Nakagomi; Tomohiro Miike; Hiroaki Shirahase; Tetsuta Oshitari; Hideyo Takahashi; Hideaki Natsugari

  CHEMISTRY-A EUROPEAN JOURNAL WILEY-V C H VERLAG GMBH 18 (6) 1572 - 1576 0947-6539 2012/02 [Refereed]
  
• B-Ring-modified and/or 5-demethylated nobiletin congeners: Inhibitory activity against pro-MMP-9 production

  Tetsuta Oshitari; Yuji Okuyama; Yoshiki Miyata; Hiroshi Kosano; Hideyo Takahashi; Hideaki Natsugari

  BIOORGANIC & MEDICINAL CHEMISTRY PERGAMON-ELSEVIER SCIENCE LTD 19 (23) 7085 - 7092 0968-0896 2011/12 [Refereed]
  
• Synthesis of New Gal beta 1 -> 4Fuc Segments Useful for Biological Investigations

  Kazusa Nishiyama; Atsushi Yamada; Tomoharu Takeuchi; Yoichiro Arata; Ken-ichi Kasai; Tetsuta Oshitari; Hideaki Natsugari; Hideyo Takahashi

  CHEMICAL & PHARMACEUTICAL BULLETIN PHARMACEUTICAL SOC JAPAN 59 (10) 1307 - 1310 0009-2363 2011/10 [Refereed]
  
• Nobiletin metabolites: Synthesis and inhibitory activity against matrix metalloproteinase-9 production

  Tetsuta Oshitari; Yuji Okuyama; Yoshiki Miyata; Hiroshi Kosano; Hideyo Takahashi; Hideaki Natsugari

  BIOORGANIC & MEDICINAL CHEMISTRY LETTERS PERGAMON-ELSEVIER SCIENCE LTD 21 (15) 4540 - 4544 0960-894X 2011/08 [Refereed]
  
• Atropisomerism Observed in Indometacin Derivatives

  Takahashi, Hideyo; Wakamatsu, Shintaro; Tabata, Hidetsugu; Oshitari, Tetsuta; Harada, Ayako; Inoue, Keizo; Natsugari, Hideaki

  ORGANIC LETTERS 13 (4) 760 - 763 2011/06 [Refereed]
  
• Isolation and Characterization of Atropisomers of Seven-Membered-Ring Benzolactams

  Hidetsugu Tabata; Naoya Wada; Yuko Takada; Tetsuta Oshitari; Hideyo Takahashi; Hideaki Natsugari

  JOURNAL OF ORGANIC CHEMISTRY AMER CHEMICAL SOC 76 (12) 5123 - 5131 0022-3263 2011/06 [Refereed]
  
• L-システイン含有アミノ酸輸液によるメロペネム水和物の分解

  工藤 千恵; 板垣 文雄; 忍足 鉄太; 高橋 秀依; 夏苅 英昭; 庭田 英明; 村上 勲; 細野 浩之; 渡邊 真知子

  日本薬学会年会要旨集 (公社)日本薬学会 131年会 (4) 252 - 252 0918-9823 2011/03
• Atropisomerism in the Vaptan Class of Vasopressin Receptor Ligands: The Active Conformation Recognized by the Receptor

  Hidetsugu Tabata; Jun Nakagomi; Daisuke Morizono; Tetsuta Oshitari; Hideyo Takahashi; Hideaki Natsugari

  ANGEWANDTE CHEMIE-INTERNATIONAL EDITION WILEY-V C H VERLAG GMBH 50 (13) 3075 - 3079 1433-7851 2011 [Refereed]
  
• Efficient Asymmetric Synthesis of Oseltamivir from D-Mannitol

  Tadakatsu Mandai; Tetsuta Oshitari

  SYNLETT GEORG THIEME VERLAG KG 2009 (5) 783 - 786 0936-5214 2009/03 [Refereed]
  
• Azide-Free Synthesis of Oseltamivir from L-Methionine

  Tetsuta Oshitari; Tadakatsu Mandai

  SYNLETT GEORG THIEME VERLAG KG 2009 (5) 787 - 789 0936-5214 2009/03 [Refereed]
  
• Asymmetric synthesis of (+)-CP-99,994 and (+)-L-733,060 from enantiomerically pure (3S,4S)-4-(tert-butylcarbamoyl)-4-phenyl-1-buten-3-ol

  Tetsuta Oshitari; Tadakatsu Mandai

  SYNLETT GEORG THIEME VERLAG KG 2006 (20) 3395 - 3398 0936-5214 2006/12 [Refereed]
  
• An efficient synthesis of optically active vicinal diamine arrays via palladium-catalyzed C-O to C-N bond transformation

  T Oshitari; R Akagi; T Mandai

  SYNTHESIS-STUTTGART GEORG THIEME VERLAG KG 2004 (9) 1325 - 1330 0039-7881 2004/06 [Refereed]
  
• A stereocontrolled synthesis of hapalosin

  T Oshitari; Saiyinbilige; T Mandai

  HETEROCYCLES PERGAMON-ELSEVIER SCIENCE LTD 62 185 - 190 0385-5414 2004/01 [Refereed]
  
• Lipase-catalyzed kinetic resolution of 4-(N-Boc-amino)-1-alken-3-ols

  T Oshitari; T Mandai

  SYNLETT GEORG THIEME VERLAG KG 2003 (15) 2374 - 2376 0936-5214 2003/12 [Refereed]
  
• Lipase-catalyzed transesterification of methyl 2-substituted 3-hydroxy-4-pentenoates and its synthetic application to the taxol side chain

  T Mandai; T Oshitari; M Susowake

  SYNLETT GEORG THIEME VERLAG KG 2002 (10) 1665 - 1668 0936-5214 2002/10 [Refereed]
  
• Synthesis and biological evaluation of water soluble taxoids bearing sugar moieties

  T Mandai; H Okumoto; T Oshitari; K Nakanishi; K Mikuni; KJ Hara; KZ Hara; W Iwatani; T Amano; K Nakamura; Y Tsuchiya

  HETEROCYCLES PERGAMON-ELSEVIER SCIENCE LTD 54 (2) 561 - + 0385-5414 2001/02 [Refereed]
  
• A practical synthetic method for alpha- and beta-glycosyloxyacetic acids

  T Mandai; H Okumoto; T Oshitari; K Nakanishi; K Mikuni; KJ Hara; KZ Hara

  HETEROCYCLES PERGAMON-ELSEVIER SCIENCE LTD 52 (1) 129 - 132 0385-5414 2000/01 [Refereed]
  
• Synthesis of 2-O-(3-O-carbamoyl-alpha-D-mannopyranosyl)-L-gulopyranose: Sugar moiety of antitumor antibiotic bleomycin

  T Oshitari; M Shibasaki; T Yoshizawa; M Tomita; K Takao; S Kobayashi

  TETRAHEDRON PERGAMON-ELSEVIER SCIENCE LTD 53 (32) 10993 - 11006 0040-4020 1997/08 [Refereed]
  
• A Synthetic Study of the Sugar Moiety of Bleomycin

  OSHITARI Tetsuta

  The University of Tokyo 1995/03 [Refereed]
  
• PREPARATION OF 2-O-(3-O-CARBAMOYL-ALPHA-D-MANNOPYRANOSYL)-L-GULOPYRANOSE - SYNTHETIC STUDY ON THE SUGAR MOIETY OF ANTITUMOR ANTIBIOTIC BLEOMYCIN

  T OSHITARI; S KOBAYASHI

  TETRAHEDRON LETTERS PERGAMON-ELSEVIER SCIENCE LTD 36 (7) 1089 - 1092 0040-4039 1995/02 [Refereed]
  
• NEW METHOD FOR THE PREPARATION OF L-GULOSE FROM D-MANNOSE - SYNTHETIC STUDY ON THE SUGAR MOIETY OF BLEOMYCIN

  T OSHITARI; M TOMITA; S KOBAYASHI

  TETRAHEDRON LETTERS PERGAMON-ELSEVIER SCIENCE LTD 35 (35) 6493 - 6494 0040-4039 1994/08 [Refereed]
  

Books etc

• 薬学演習Ⅱ 基礎科学

  日本薬学会 (問8・54〜8・68、11・32、11・34、11・36、11・38、11・40、11・42、Act30,31)東京化学同人 2021/10 9784807917242 xii, 493p
• ブランニューアプローチ新釈薬理論 : 受容体から生体,疾患,そして薬の関係を考える

  小野, 景義; 忍足, 鉄太 京都廣川書店 2021/03 9784909197818 xi, 575p
• 知っておきたい有機反応100 第２版

  日本薬学会編 (Joint work第XIII部 還元反応)東京化学同人 2019/03 9784807909605 290 228-241
• ベーシック薬学教科書シリーズ ５ 有機化学 第２版

  夏苅; 高橋編; 東屋、赤井; 岩渕; 忍足; 白井; 杉原; 田村 (Joint work17章 炭素骨格を構築する合成反応と官能基変換)化学同人 2016/04 9784759816228 447 345-368
• スタンダード薬学シリーズ II 3 化学系薬学 II. 生体分子・医薬品の化学による理解

  日本薬学会編 (Joint work第11章 酵素に作用する医薬品の構造と性質 SBO28, 29)東京化学同人 2016/03 9784807917068 346 232-243
• ベーシック薬学教科書シリーズ５ 有機化学

  OSHITARI Tetsuta (Joint workChapter 17)化学同人 2008/12 9784759812558 447 369-395

MISC

• Membrane permeability of diphenhydramine derivatives via H⁺/organic cation antiporter

  手賀悠真; 田畑英嗣; 黒澤俊樹; 北村敦; 板垣文雄; 忍足鉄太; 出口芳春  日本薬学会年会要旨集(CD-ROM)  140th-  2020
• ヒト血液脳関門におけるH⁺/有機カチオン交換輸送体の基質認識性についての検討

  手賀悠真; 田畑英嗣; 黒澤俊樹; 北村敦; 板垣文雄; 忍足鉄太; 出口芳春  日本薬剤学会年会講演要旨集(Web)  34th-  2019
• 血液脳関門におけるH⁺/有機カチオン交換輸送体を介した輸送への化学構造の影響

  手賀悠真; 田畑英嗣; 黒澤俊樹; 北村敦; 板垣文雄; 忍足鉄太; 出口芳春  生体膜と薬物の相互作用シンポジウム講演要旨集  41st-  2019
• ヒト血液脳関門におけるH⁺/有機カチオン交換輸送体の基質探索研究

  手賀悠真; 田畑英嗣; 黒澤俊樹; 北村敦; 板垣文雄; 忍足鉄太; 出口芳春  日本薬学会関東支部大会講演要旨集  63rd-  2019
• 合成カンナビノイド誘導体の合成とGC-MS/MSによる位置異性体識別

  荒木拡嗣; 牧野宏章; 松本謙吾; 草野麻衣子; 財津桂; 田畑英嗣; 忍足鉄太; 夏苅英昭; 高橋秀依  日本薬学会関東支部大会講演要旨集  62nd-  2018
• カルバペネム系抗生物質とL-システインの配合変化物における細胞生存率への影響

  中川 幸子; 板垣 文雄; 飯島 亮介; 忍足 鉄太; 高橋 秀依; 夏苅 英昭; 油井 聡; 鈴木 るね; 関谷 朱美; 西 優; 山元 孝俊; 渡邊 真知子  医療薬学フォーラム2014/第22回クリニカルファーマシーシンポジウム抄録集  2014/06
• Book review

  OSHITARI Tetsuta  Chemistry  69-  (2)  56  -56  2014/02  [Invited]
  
• フッ素を含有した新規リン脂質の開発

  森達也; 小田雄介; 宇留賀仁史; 鈴木亮; 丸山一雄; 忍足鉄太; 夏苅英昭; 高橋秀依  日本薬学会年会要旨集(CD-ROM)  134th-  2014
• 銅-ジスルフィラム錯体の可溶化

  星佑次郎; 谷紀彦; 田畑英嗣; 関むつみ; 鈴木亮; 丸山一雄; 宗形光敏; 児玉浩子; 忍足鉄太; 夏苅英昭; 高橋秀依  日本薬学会年会要旨集(CD-ROM)  134th-  2014
• メロペネムとSH基を有する医薬品の配合変化

  片桐幸子; 板垣文雄; 忍足鉄太; 高橋秀依; 夏苅英昭; 渡邊真知子  日本薬学会年会要旨集(CD-ROM)  133rd-  (4)  ROMBUNNO.29PMF-382  -152  2013
• L‐システインによるβ‐ラクタム系抗生物質の分解

  片桐幸子; 工藤千恵; 板垣文雄; 忍足鉄太; 高橋秀依; 夏苅英昭; 庭田英明; 渡邊真知子  日本医療薬学会年会講演要旨集  22nd-  345  2012/10
• P2-144 L-システインはメロペネム水和物のβ-ラクタム環を開環して配合変化を惹き起す(一般演題 ポスター発表,薬物相互作用,臨床から学び臨床へと還元する医療薬学)

  工藤 千恵; 板垣 文雄; 忍足 鉄太; 高橋 秀依; 夏苅 英昭; 庭田 英明; 村上 勲; 細野 浩之; 渡邊 真知子  日本医療薬学会年会講演要旨集  20-  414  -414  2010/10
• A new synthetic method for chiral 1,2-diamines and its application to the synthesis of bioactive piperidine derivatives

  Tetsuta Oshitari; Tadakatsu Mandai  JOURNAL OF MOLECULAR CATALYSIS B-ENZYMATIC  48-  (3-4)  112  -113  2007/09
• Lipase-catalyzed transesterification of methyl 2-substituted 3-hydroxy-4-pentenoates and its synthetic application to the taxol side chain

  T Mandai; T Oshitari; M Susowake  SYNLETT  2002-  (10)  1665  -1668  2002/10
• Creation of non-peptide aspartic peptidase inhibitors.

  OSHITARI Tetsuta  Farumashia  38-  (4)  338  -339  2002  [Invited]
  
• Synthesis and biological evaluation of water soluble taxoids bearing sugar moieties

  T Mandai; H Okumoto; T Oshitari; K Nakanishi; K Mikuni; KJ Hara; KZ Hara; W Iwatani; T Amano; K Nakamura; Y Tsuchiya  HETEROCYCLES  54-  (2)  561  -+  2001/02
• A practical synthetic method for alpha- and beta-glycosyloxyacetic acids

  T Mandai; H Okumoto; T Oshitari; K Nakanishi; K Mikuni; KJ Hara; KZ Hara  HETEROCYCLES  52-  (1)  129  -132  2000/01

Research Grants & Projects

• Search and application of novel functional food and its components that prevent thrombosis caused by modern lifestyle

  Japan Society for the Promotion of Science：Grants-in-Aid for Scientific Research

  Date (from‐to) : 2016/04 -2019/03 

  Author : Naoki Ohkura
• 多機能なポリメトキシフラボン類の活性分離と標的への送達を指向した合成戦略の展開

  独立行政法人日本学術振興会：学術研究助成基金助成金（基盤研究（Ｃ））

  Date (from‐to) : 2015/04 -2017/03 

  Author : 忍足 鉄太
• Exploration of antithrombotic substanse and development of new functional foods that prevent aging induced thrombotic conditions

  Japan Society for the Promotion of Science：Grants-in-Aid for Scientific Research

  Date (from‐to) : 2013/04 -2016/03 

  Author : Ohkura Naoki; Oishi KATSUTAKA; ATSUMI GEN-ICHI; OSHITARI TETSUTA; TANIGUCHI MASAHIKO
• Prevention research for diabetic retinopathy based on structure-activity relationship study of novel polymethoxyflavones

  Japan Society for the Promotion of Science：Grants-in-Aid for Scientific Research

  Date (from‐to) : 2013/04 -2015/03 

  Author : MIYATA Yoshiki; OSHITARI Tetsuta
• 水溶性タキソ-ル誘導体の合成研究

  日本学術振興会：科学研究費助成事業

  Date (from‐to) : 1997 -1997 

  Author : 萬代 忠勝; 忍足 鉄太
• 水溶性タキソ-ル誘導体の合成研究

  日本学術振興会：科学研究費助成事業

  Date (from‐to) : 1996 -1996 

  Author : 萬代 忠勝; 忍足 鉄太
• Organometallic Chemistry
• Synthetic Study of Bioactive Compounds